Active Substance: Exemestane
Packaging: 30*25mg tablets
Exemastane is an aromatize inhibitor and used in steroid cycles or TRT (Testosterone Replacement Therapy)
Exemestane by Actavis
Exemestane is one of the aromatase inhibitors of the third Generation and was developed as any other aromatase inhibitor for the treatment of estrogen- induced breast cancer in women.
Unlike older aromatase inhibitors exemestan docked firmly to the aromatase enzyme and this may disable permanently so . This connection can be released again , so that the aromatase enzyme is then re- activated .
In bodybuilding exemestan finds its application to the side-effects of anabolic and androgenic steroids Down to suppress . The flavoring by anabolic steroid abuse are bound by the drug exemestan for the most part .
Exemestane contains a very efficient aromatase . The activity of the enzyme aromatase is suppressed by up to 98 %, which means a reduction in the estrogen levels by 85 %. In comparison, the reduction in estrogen aromatase inhibitors such as anastrozole is at or letrozole in just under 80 %. For this reason, exemestan is the most valued among bodybuilders aromatase .
In this context, is to note that estrogen also has some anabolic effect and a strong reduction in estrogen levels through the use of aromatase inhibitors such as exemestan during use of anabolic androgenic steroids can result in reduced gains in muscle mass .
Side effects :
Hot flashes, nausea, fatigue, sweating, headache, insomnia, depression, decrease in lymphocytes, thrombocytopenia, leukopenia, elevation of liver enzymes, hypertrichosis, hair loss, hoarseness, acne
Application / dosage :
In bodybuilding, the half a tablet (12.5 mg exemestane) is usually used every day, or every 2 days one tablet ( 25mg exemestane) . in the last phase of a pre-contest bodybuilders take some daily 25mg exemestane .
Optimal is a intake after a high fat meal, because as the bioavailability can be increased by up to 40 percent. Until when taking exemestane stable blood levels are reached , passing by the manufacturer about a week.